Lidanserin
Lidanserin (INN; ZK-33,839) is a drug which acts as a combined 5-HT2A and α1-adrenergic receptor antagonist.[1] It was developed as an antihypertensive agent but was never marketed.[1]
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Formula | C26H31FN2O4 |
Molar mass | 454.542 g·mol−1 |
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References
- Allen RC (1989). Annual Reports in Medicinal Chemistry. Academic Press. p. 56. ISBN 978-0-12-040524-4. Retrieved 6 May 2012.
Sympatholytics (antagonize α-adrenergic vasoconstriction) | |||||
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α1 |
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α2 |
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β |
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5-HT1 |
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5-HT2 |
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5-HT3–7 |
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