Testosterone nicotinate

Testosterone nicotinate (brand names Bolfortan, Linobol) is an androgen and anabolic steroid medication made by esterifying nicotinic acid and testosterone[1][2][3][4][5] It was formulated as a 50 mg/mL aqueous suspension provided in ampoules.[4][5] The medication was manufactured and sold by Lannacher Heilmittel GmbH in Austria.[5] It is no longer marketed.[5]

Testosterone nicotinate
Clinical data
Trade namesBolfortan, Linobol
Other namesWD-53
Routes of
administration
Intramuscular injection
Identifiers
IUPAC name
  • (1S,2R,10R,11S,14S,15S)-2,15-dimethyl-5-oxotetracyclo[8.7.0.02,7.011,15]heptadec-6-en-14-yl pyridine-3-carboxylate
CAS Number
PubChem CID
ChemSpider
UNII
CompTox Dashboard (EPA)
ECHA InfoCard100.010.522
Chemical and physical data
FormulaC25H31NO3
Molar mass393.527 g·mol−1
3D model (JSmol)
SMILES
  • C[C@]12CC[C@H]3[C@H]([C@@H]1CC[C@@H]2OC(=O)C4=CN=CC=C4)CCC5=CC(=O)CC[C@]35C
InChI
  • InChI=1S/C25H31NO3/c1-24-11-9-18(27)14-17(24)5-6-19-20-7-8-22(25(20,2)12-10-21(19)24)29-23(28)16-4-3-13-26-15-16/h3-4,13-15,19-22H,5-12H2,1-2H3/t19-,20-,21-,22-,24-,25-/m0/s1
  • Key:KHRRLLSDLVLEIT-BKWLFHPQSA-N

Testosterone nicotinate had a relatively short duration, somewhere between that of testosterone propionate and testosterone enanthate.[5][4]

See also

References

  1. Elks J (14 November 2014). The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. pp. 641–642. ISBN 978-1-4757-2085-3.
  2. Index Nominum 2000: International Drug Directory. Taylor & Francis. January 2000. ISBN 978-3-88763-075-1.
  3. Morton IK, Hall JM (6 December 2012). Concise Dictionary of Pharmacological Agents: Properties and Synonyms. Springer Science & Business Media. ISBN 978-94-011-4439-1.
  4. Virginia. Task Force on Anabolic Steroid Misuse Among Minors (1988). Report of the Task Force on Anabolic Steroid Misuse Among Minors: To the Director, Virginia Department of Health Regulatory Boards. Department of Health Regulatory Boards. BOLFORTAN injection 50mgs/cc 1 ampules Lanniker Heilmittel, Austria cc Bolfortan is an nicotinate. The nicotinate added to the steroid molecule makes it last longer than regular [...] make this short, aqueous testosterone testosterone aqueous, although being water based, this form of testosterone gets into the system rather quickly. Testosterone Nicotinate has a half-life somewhere between Testosterone Propionate and Testosterone Enanthate.
  5. Llewellyn W (2011). Anabolics. Molecular Nutrition LLC. pp. 182–184. ISBN 978-0-9828280-1-4.



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