Properidine

Properidine is an opioid, an analgesic, and the isopropyl analog of pethidine.[1] Properidine is under international control and is listed in the United States under the Controlled Substances Act (1970) as a Schedule I substance. It is a narcotic, with an Administrative Controlled Substances Code Number (ACSCN) of 9644 and a 2 gramme annual aggregate manufacturing quota as of 2014. The salt in use is hydrochloride, with a free base conversion ratio of 0.88.[2]

Properidine
Clinical data
Other namesIpropethidine
ATC code
  • none
Legal status
Legal status
  • AU: S9 (Prohibited substance)
  • CA: Schedule I
  • DE: Anlage I (Authorized scientific use only)
  • UK: Class A
  • US: Schedule I
  • UN: Psychotropic Schedule I
Identifiers
IUPAC name
  • isopropyl 1-methyl-4-phenylpiperidine-4-carboxylate
CAS Number
PubChem CID
ChemSpider
UNII
CompTox Dashboard (EPA)
ECHA InfoCard100.008.385
Chemical and physical data
FormulaC16H23NO2
Molar mass261.365 g·mol−1
3D model (JSmol)
SMILES
  • O=C(OC(C)C)C2(c1ccccc1)CCN(C)CC2
InChI
  • InChI=1S/C16H23NO2/c1-13(2)19-15(18)16(9-11-17(3)12-10-16)14-7-5-4-6-8-14/h4-8,13H,9-12H2,1-3H3 Y
  • Key:XJKQCILVUHXVIQ-UHFFFAOYSA-N Y
 NY (what is this?)  (verify)

References
  1. Morrison AL, Rinderknecht H (1950). "302. Synthetic analgesics. Part V. Compounds related to pethidine". Journal of the Chemical Society (Resumed): 1467. doi:10.1039/JR9500001467.
  2. "Quotas - 2014". Diversion Control Division. U.S. Department of Justice, Drug Enforcement Administration.


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