Methimepip

Methimepip
Names
	IUPAC name 4-(1H-imidazol-4-ylmethyl)-1-methylpiperidine
Identifiers
CAS Number	151070-80-3 ;
3D model (JSmol)	Interactive image;
ChEMBL	ChEMBL175782 ;
ChemSpider	9488804 ;
IUPHAR/BPS	1254;
MeSH	C500075
PubChem CID	11313837;
CompTox Dashboard (EPA)	DTXSID80462102 ;
	InChI InChI=1S/C10H17N3/c1-13-4-2-9(3-5-13)6-10-7-11-8-12-10/h7-9H,2-6H2,1H3,(H,11,12) Key: KIAVPENCSGKVQP-UHFFFAOYSA-N ; InChI=1/C10H17N3/c1-13-4-2-9(3-5-13)6-10-7-11-8-12-10/h7-9H,2-6H2,1H3,(H,11,12) Key: KIAVPENCSGKVQP-UHFFFAOYAQ;
	SMILES CN1CCC(CC1)CC2=CN=CN2;
Properties
Chemical formula	C10H17N3
Molar mass	179.262 g/mol
	Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
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	Infobox references

Methimepip is a histamine agonist which is highly selective for the H₃ subtype. It is the N-methyl derivative of immepip.^[1]

References

↑ Kitbunnadaj R, Hashimoto T, Poli E, et al. (March 2005). "N-substituted piperidinyl alkyl imidazoles: discovery of methimepip as a potent and selective histamine H3 receptor agonist". Journal of Medicinal Chemistry. 48 (6): 2100–7. doi:10.1021/jm049475h. PMID 15771452.

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