O-4310

O-4310
Identifiers
IUPAC name
  • 3-[2-(dimethylamino)ethyl]-6-fluoro-1-isopropyl-1H-indol-4-ol
CAS Number
PubChem CID
UNII
Chemical and physical data
FormulaC15H21FN2O
Molar mass264.344 g·mol−1
3D model (JSmol)
SMILES
  • CC(C)N1C2=CC(F)=CC(O)=C2C(CCN(C)C)=C1

O-4310 (1-isopropyl-6-fluoro-psilocin) is a tryptamine derivative developed by Organix Inc which acts as a serotonin receptor agonist. It is claimed to have an EC50 of 5nM at 5-HT2A with 89% efficacy vs 5-HT, and 100x selectivity over 5-HT2C, while being apparently inactive at the 5-HT2B antitarget.[1]

See also

References

  1. ↑ US 7655691, Kumaran G, Morency C, Roth B, Sard HP, Shuster L, Xu L, "Indole compounds useful as serotonin selective agents.", published 11 May 2006, assigned to Organix Inc


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