Ebalzotan
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| Routes of administration | Oral |
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IUPAC name
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| Formula | C19H30N2O2 |
| Molar mass | 318.461 g·mol−1 |
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Ebalzotan (NAE-086) is a selective 5-HT1A receptor agonist.[1][2] It was under development as an antidepressant and anxiolytic agent but produced undesirable side effects in phase I clinical trials and was subsequently discontinued.[1][2]
See also
References
- 1 2 Braish T, Gadamasetti KG (2008). Process chemistry in the pharmaceutical industry, volume 2 challenges in an ever changing climate. Boca Raton: CRC Press. ISBN 978-0-8493-9051-7.
- 1 2 Weaver DF, Nogrady T, Nogrady T (2005). Medicinal chemistry a molecular and biochemical approach. Oxford [Oxfordshire]: Oxford University Press. ISBN 0-19-510455-2.
| 5-HT1AR agonists | |
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| GABAAR PAMs |
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| Gabapentinoids (α2δ VDCC blockers) | |
| Antidepressants |
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| Sympatholytics (Antiadrenergics) |
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Serotonin receptor modulators | |||||||||||||||||||||||||||||||||||||||
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| 5-HT1 |
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| 5-HT2 |
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| 5-HT3–7 |
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