Profadol

Profadol
Clinical data
ATC code
  • none
Legal status
Legal status
Identifiers
IUPAC name
  • 3-(1-methyl-3-propyl-pyrrolidin-3-yl)phenol
CAS Number
PubChem CID
ChemSpider
UNII
ChEMBL
Chemical and physical data
FormulaC14H21NO
Molar mass219.328 g·mol−1

Profadol (CI-572) is an opioid analgesic which was developed in the 1960s by Parke-Davis.[1] It acts as a mixed agonist-antagonist of the μ-opioid receptor. The analgetic potency is about the same as of pethidine (meperidine), the antagonistic effect is 1/50 of nalorphine.[2]

See also

References

  1. DE 1303096
  2. Schröder E, Rufer C, Schmiechen R (1976). Arzneimittelchemie 1. Grundlagen, Nerven, Muskeln und Gewebe. Stuttgart: Georg Thieme Verlag. ISBN 3-13-520601-7.
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