Cyprodenate

Cyprodenate (Actebral) is a stimulant drug.[1] It was used for counteracting the effects of benzodiazepine tranquillizer drugs before the development of newer antidotes such as flumazenil.[2] It produces dimethylethanolamine as a metabolite.

Cyprodenate
Clinical data
AHFS/Drugs.comInternational Drug Names
ATC code
  • N06BX04
Identifiers
IUPAC name
  • 2-dimethylaminoethyl 3-cyclohexylpropanoate
CAS Number
PubChem CID
ChemSpider
UNII
KEGG
ChEMBL
CompTox Dashboard (EPA)
ECHA InfoCard100.036.025
Chemical and physical data
FormulaC13H25NO2
Molar mass227.34 g·mol−1
3D model (JSmol)
SMILES
  • CN(C)CCOC(=O)CCC1CCCCC1
InChI
  • InChI=1S/C13H25NO2/c1-14(2)10-11-16-13(15)9-8-12-6-4-3-5-7-12/h12H,3-11H2,1-2H3 Y
  • Key:MPOYJPINNSIHAK-UHFFFAOYSA-N Y
  (verify)

See also

References
  1. Dormard Y, Levron JC, Le Fur JM (February 1975). "Pharmacokinetic study of maleate acid of 2-(N,N-dimethylaminoethanol-14C1)-cyclohexylpropionate (cyprodenate) and of N,N-dimethylaminoethanol-14C1 in animals". Arzneimittel-Forschung. 25 (2): 201–7. PMID 1173033.
  2. Bobkov I, Morozov IS (October 1982). "[Correction of psychodepressive effects of benzodiazepine tranquilizers by administration of psychostimulants]". Biulleten' Eksperimental'noi Biologii I Meditsiny. 94 (10): 48–51. doi:10.1007/BF00827201. PMID 6129008. S2CID 19153614.


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