Pelanserin

Pelanserin
Names
	Preferred IUPAC name 3-[3-(4-Phenylpiperazin-1-yl)propyl]quinazoline-2,4(1H,3H)-dione
Identifiers
CAS Number	2208-51-7 ;
3D model (JSmol)	Interactive image;
ChemSpider	58898;
PubChem CID	65435;
UNII	6SNR96E409 ;
CompTox Dashboard (EPA)	DTXSID60176578 ;
	InChI InChI=1S/C21H24N4O2/c26-20-18-9-4-5-10-19(18)22-21(27)25(20)12-6-11-23-13-15-24(16-14-23)17-7-2-1-3-8-17/h1-5,7-10H,6,11-16H2,(H,22,27) Key: WPKPLSFHHBBLRY-UHFFFAOYSA-N; InChI=1/C21H24N4O2/c26-20-18-9-4-5-10-19(18)22-21(27)25(20)12-6-11-23-13-15-24(16-14-23)17-7-2-1-3-8-17/h1-5,7-10H,6,11-16H2,(H,22,27) Key: WPKPLSFHHBBLRY-UHFFFAOYAV;
	SMILES C1CN(CCN1CCCN2C(=O)C3=CC=CC=C3NC2=O)C4=CC=CC=C4;
Properties
Chemical formula	C21H24N4O2
Molar mass	364.449 g·mol−1
	Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa). Infobox references

Pelanserin is an antagonist of the 5-HT₂ and α₁-adrenergic receptors.[1]

References

Villalobos-Molina, R; Ibarra, M; Hong, E (1995). "The 5-HT2 receptor antagonist, pelanserin, inhibits alpha 1-adrenoceptor-mediated vasoconstriction in vitro". European Journal of Pharmacology. 277 (2–3): 181–5. doi:10.1016/0014-2999(95)00074-u. PMID 7493607.

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