Barbexaclone
Barbexaclone (Maliasin) is a salt compound of phenobarbital and levopropylhexedrine.[1] It was introduced in 1983. It has been reported to be as effective as phenobarbital but better tolerated; however, as of 2004, these "promising results"[2] had not yet been confirmed nor denied in controlled trials.
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Phenobarbital | Barbiturate |
Levopropylhexedrine | Stimulant (sympathomimetic) |
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ECHA InfoCard | 100.022.278 |
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Potency
100 mg of barbexaclone is equivalent to 60 mg of phenobarbital.[1]
References
- Shorvon S, Perucca E, Engel Jr J (23 September 2015). The Treatment of Epilepsy. Wiley. pp. 1706–1707. ISBN 978-1-118-93699-3.
- Salles Barbosa MF (September 1978). "[Barbexaclone in the treatment of cerebral dysrhythmia]". Arquivos de Neuro-Psiquiatria. 36 (3): 245–9. doi:10.1590/s0004-282x1978000300009. PMID 28716.
Further reading
- Shorvon SR, Fish DR, Perucca E, Dodson WE, eds. (2004). The Treatment of Epilepsy (2nd ed.). Published by Blackwell. p. 472. ISBN 0-632-06046-8.
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See also: Receptor/signaling modulators • GABA receptor modulators • GABA metabolism/transport modulators |
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